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Calcium in PDB 3iit: Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane DerivativeEnzymatic activity of Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative
All present enzymatic activity of Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative:
3.4.21.6; Protein crystallography data
The structure of Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative, PDB code: 3iit
was solved by
M.Suzuki,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 3iit:
The structure of Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative also contains other interesting chemical elements:
Calcium Binding Sites:
The binding sites of Calcium atom in the Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative
(pdb code 3iit). This binding sites where shown within
5.0 Angstroms radius around Calcium atom.
In total 2 binding sites of Calcium where determined in the Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative, PDB code: 3iit: Jump to Calcium binding site number: 1; 2; Calcium binding site 1 out of 2 in 3iitGo back to Calcium Binding Sites List in 3iit
Calcium binding site 1 out
of 2 in the Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative
Mono view Stereo pair view
Calcium binding site 2 out of 2 in 3iitGo back to Calcium Binding Sites List in 3iit
Calcium binding site 2 out
of 2 in the Factor Xa in Complex with A Cis-1,2-Diaminocyclohexane Derivative
Mono view Stereo pair view
Reference:
K.Yoshikawa,
S.Kobayashi,
Y.Nakamoto,
N.Haginoya,
S.Komoriya,
T.Yoshino,
T.Nagata,
A.Mochizuki,
K.Watanabe,
M.Suzuki,
H.Kanno,
T.Ohta.
Design, Synthesis, and Sar of Cis-1,2-Diaminocyclohexane Derivatives As Potent Factor Xa Inhibitors. Part II: Exploration of 6-6 Fused Rings As Alternative S1 Moieties. Bioorg.Med.Chem. V. 17 8221 2009.
Page generated: Sat Dec 12 04:15:30 2020
ISSN: ISSN 0968-0896 PubMed: 19900814 DOI: 10.1016/J.BMC.2009.10.024 |
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