|
Atomistry » Calcium » PDB 2wuv-2xc4 » 2xbx | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Calcium » PDB 2wuv-2xc4 » 2xbx » |
Calcium in PDB 2xbx: Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid InhibitorEnzymatic activity of Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor
All present enzymatic activity of Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor:
3.4.21.6; Protein crystallography data
The structure of Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor, PDB code: 2xbx
was solved by
D.W.Banner,
J.Benz,
D.Schlatter,
W.Haap,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 2xbx:
The structure of Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor also contains other interesting chemical elements:
Calcium Binding Sites:
The binding sites of Calcium atom in the Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor
(pdb code 2xbx). This binding sites where shown within
5.0 Angstroms radius around Calcium atom.
In total only one binding site of Calcium was determined in the Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor, PDB code: 2xbx: Calcium binding site 1 out of 1 in 2xbxGo back to![]() ![]()
Calcium binding site 1 out
of 1 in the Factor Xa in Complex with A Pyrrolidine-3,4-Dicarboxylic Acid Inhibitor
![]() Mono view ![]() Stereo pair view
Reference:
L.Anselm,
D.W.Banner,
J.Benz,
K.Groebke Zbinden,
J.Himber,
H.Hilpert,
W.Huber,
B.Kuhn,
J.L.Mary,
M.B.Otteneder,
N.Panday,
F.Ricklin,
M.Stahl,
S.Thomi,
W.Haap.
Discovery of A Factor Xa Inhibitor (3R,4R)-1-(2,2-Difluoro-Ethyl)-Pyrrolidine-3,4-Dicarboxylic Acid 3-[(5-Chloro-Pyridin-2-Yl)-Amide] 4-{[2-Fluoro-4-(2-Oxo-2H-Pyridin-1-Yl)-Phenyl]-Amide} As A Clinical Candidate. Bioorg.Med.Chem. V. 20 5313 2010.
Page generated: Tue Jul 8 09:20:01 2025
ISSN: ISSN 0968-0896 PubMed: 20650636 DOI: 10.1016/J.BMCL.2010.06.126 |
Last articlesMg in 3D2JMg in 3D2E Mg in 3D1R Mg in 3CXC Mg in 3CPW Mg in 3CZJ Mg in 3D19 Mg in 3CZ4 Mg in 3CZ1 Mg in 3CZ0 |
© Copyright 2008-2020 by atomistry.com | ||
Home | Site Map | Copyright | Contact us | Privacy |