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Atomistry » Calcium » PDB 5agv-5b4y » 5ar5 » |
Calcium in PDB 5ar5: RIP2 Kinase Catalytic Domain (1 - 310) Complex with BenzimidazoleEnzymatic activity of RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole
All present enzymatic activity of RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole:
2.7.10.2; 2.7.11.1; Protein crystallography data
The structure of RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole, PDB code: 5ar5
was solved by
A.K.Charnley,
M.A.Convery,
A.Lakdawala Shah,
E.Jones,
P.Hardwicke,
A.Bridges,
B.J.Votta,
P.J.Gough,
R.W.Marquis,
J.Bertin,
L.Casillas,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 5ar5:
The structure of RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole also contains other interesting chemical elements:
Calcium Binding Sites:
The binding sites of Calcium atom in the RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole
(pdb code 5ar5). This binding sites where shown within
5.0 Angstroms radius around Calcium atom.
In total only one binding site of Calcium was determined in the RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole, PDB code: 5ar5: Calcium binding site 1 out of 1 in 5ar5Go back to![]() ![]()
Calcium binding site 1 out
of 1 in the RIP2 Kinase Catalytic Domain (1 - 310) Complex with Benzimidazole
![]() Mono view ![]() Stereo pair view
Reference:
A.K.Charnley,
M.A.Convery,
A.Lakdawala Shah,
E.Jones,
P.Hardwicke,
A.Bridges,
M.Ouellette,
R.Totoritis,
B.Schwartz,
B.W.King,
D.D.Wisnoski,
J.Kang,
P.M.Eidam,
B.J.Votta,
P.J.Gough,
R.W.Marquis,
J.Bertin,
L.Casillas.
Crystal Structures of Human RIP2 Kinase Catalytic Domain Complexed with Atp-Competitive Inhibitors: Foundations For Understanding Inhibitor Selectivity. Bioorg.Med.Chem. V. 23 7000 2015.
Page generated: Sun Jul 14 16:37:06 2024
ISSN: ISSN 0968-0896 PubMed: 26455654 DOI: 10.1016/J.BMC.2015.09.038 |
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